Tham khảo L-655,708

  1. Quirk, K; Blurton, P; Fletcher, S; Leeson, P; Tang, F; Mellilo, D; Ragan, CI; McKernan, RM (1996). “3HL-655,708, a novel ligand selective for the benzodiazepine site of GABAA receptors which contain the alpha 5 subunit”. Neuropharmacology. 35 (9–10): 1331–5. doi:10.1016/S0028-3908(96)00061-5. PMID 9014149.
  2. Casula, MA; Bromidge, FA; Pillai, GV; Wingrove, PB; Martin, K; Maubach, K; Seabrook, GR; Whiting, PJ; Hadingham, KL (2001). “Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor”. Journal of Neurochemistry. 77 (2): 445–51. doi:10.1046/j.1471-4159.2001.00289.x. PMID 11299307.
  3. Sur, C; Fresu, L; Howell, O; McKernan, RM; Atack, JR (1999). “Autoradiographic localization of alpha5 subunit-containing GABAA receptors in rat brain”. Brain Research. 822 (1–2): 265–70. doi:10.1016/S0006-8993(99)01152-X. PMID 10082908.
  4. Chambers, MS; Atack, JR; Broughton, HB; Collinson, N; Cook, S; Dawson, GR; Hobbs, SC; Marshall, G; Maubach, KA (2003). “Identification of a novel, selective GABA(A) alpha5 receptor inverse agonist which enhances cognition”. Journal of Medicinal Chemistry. 46 (11): 2227–40. doi:10.1021/jm020582q. PMID 12747794. Đã bỏ qua tham số không rõ |displayauthors= (gợi ý |display-authors=) (trợ giúp)
  5. Chambers, MS; Atack, JR; Carling, RW; Collinson, N; Cook, SM; Dawson, GR; Ferris, P; Hobbs, SC; O'Connor, D (2004). “An orally bioavailable, functionally selective inverse agonist at the benzodiazepine site of GABAA alpha5 receptors with cognition enhancing properties”. Journal of Medicinal Chemistry. 47 (24): 5829–32. doi:10.1021/jm040863t. PMID 15537339. Đã bỏ qua tham số không rõ |displayauthors= (gợi ý |display-authors=) (trợ giúp)
  6. Atack, JR; Bayley, PJ; Seabrook, GR; Wafford, KA; McKernan, RM; Dawson, GR (2006). “L-655,708 enhances cognition in rats but is not proconvulsant at a dose selective for alpha5-containing GABAA receptors”. Neuropharmacology. 51 (6): 1023–9. doi:10.1016/j.neuropharm.2006.04.018. PMID 17046030.
  7. Navarro, JF; Burón, E; Martín-López, M (2002). “Anxiogenic-like activity of L-655,708, a selective ligand for the benzodiazepine site of GABA(A) receptors which contain the alpha-5 subunit, in the elevated plus-maze test”. Progress in Neuro-Psychopharmacology & Biological Psychiatry. 26 (7–8): 1389–92. doi:10.1016/S0278-5846(02)00305-6. PMID 12502028.
  8. Saab, BJ; Maclean AJ; Kanisek M; Zurek AA; Martin LJ; Roder JC; Orser BA (tháng 11 năm 2010). “Short-term memory impairment after isoflurane in mice is prevented by the α5 γ-aminobutyric acid type A receptor inverse agonist L-655,708”. Anesthesiology. 113 (5): 1061–71. doi:10.1097/ALN.0b013e3181f56228. PMID 20966663.
  9. Fischell, Jonathan; Van Dyke, Adam M; Kvarta, Mark D; LeGates, Tara A; Thompson, Scott M (2015). “Rapid Antidepressant Action and Restoration of Excitatory Synaptic Strength After Chronic Stress by Negative Modulators of Alpha5-Containing GABAA Receptors”. Neuropsychopharmacology. 40: 2499–2509. doi:10.1038/npp.2015.112. ISSN 0893-133X. PMC 4569955. PMID 25900119.

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